Skip to main content

Table 1 The cocktail probe of different concentration (μM)

From: Triptolide Induces hepatotoxicity via inhibition of CYP450s in Rat liver microsomes

Substrates

Concentration Number

1

2

3

4

5

6

7

Caffeine(CAF)

1.875

3.75

7.5

15

30

60

120

Tolbutamide(D860)

0.625

1.25

2.5

5

10

20

40

(S)- Mephenytoin(MT)

1.25

2.5

5

10

20

40

60

Dextromethorphan(DM)

2.5

5

10

20

40

80

160

Chlorzoxazone(CLZ)

1.25

2.5

5

10

20

40

60

Midazolam(MDZ)

0.313

0.625

1.25

2.5

5

10

20